SCHEMBL28447722

SCHEMBL28447722

C=CC(=O)Nc1ccc(OC)c(Nc2nccc(Nc3ccc(N4CCOCC4)cc3OC)n2)c1

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.78
JAK3 P52333 1/20 0.62
ALK Q9UM73 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053852 0.91 EGFR (0.78) EGFRJAK3ALK
SCHEMBL28053996 0.90 ALK (0.75) EGFRJAK3ALK
SCHEMBL28452560 0.88 EGFR (0.73) EGFRJAK3ALK
SCHEMBL17059584 0.88 EGFR (1.00) EGFRJAK3
SCHEMBL28053999 0.87 EGFR (0.65) EGFRJAK3ALK
SCHEMBL28053986 0.87 EGFR (0.80) EGFRJAK3ALK
SCHEMBL28053865 0.87 EGFR (0.83) EGFRJAK3ALK
Hydrochloric Acid SCHEMBL28053870 0.86 EGFR (0.82) EGFRJAK3ALK
SCHEMBL17059625 0.83 EGFR (1.00) EGFRJAK3
SCHEMBL28915867 0.81 EGFR (0.75) EGFRJAK3ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed