SCHEMBL28055137

SCHEMBL28055137

C[C@@H]1NCCN(CCCCC(=O)OC(C)(C)C)C1=O.O=COCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.42
PLA2G5 P39877 1/20 0.42
FAAH O00519 4/20 0.36
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 2/20 0.35
CYP3A4 P08684 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PKM P14618 2/20 0.35
GAA P10253 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
CTSL P07711 1/20 0.34
TSHR P16473 4/20 0.34
MAPK1 P28482 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28055093 0.97 PLA2G10 (0.42) PLA2G10PLA2G5FAAHALDH1A1KDM4E
SCHEMBL27894045 0.94 PLA2G10 (0.43) PLA2G10PLA2G5FAAHMEN1KMT2A
SCHEMBL28055160 0.89 TSHR (0.42) ALDH1A1KDM4EMEN1LMNACYP3A4
SCHEMBL1586934 0.82 PLA2G10 (0.39) PLA2G10PLA2G5
SCHEMBL1554996 0.82 PLA2G10 (0.39) PLA2G10PLA2G5
SCHEMBL27894049 0.80 PKM (0.38) PLA2G10PLA2G5MEN1KMT2ASMN1; SMN2
SCHEMBL1556365 0.78 PLA2G10 (0.40) PLA2G10PLA2G5
SCHEMBL1555754 0.78 PLA2G10 (0.40) PLA2G10PLA2G5
SCHEMBL1586781 0.75 PDK1 (0.43) ALDH1A1
SCHEMBL1555362 0.75 PDK1 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102762541-B Diaza derivatives as modulators of chemokine receptors HOFFMAN-LA ROCHE LTD. (CH) 2016-03-16 CN disclosed
CN-102762541-A Diaza derivatives as modulators of chemokine receptors HOFFMANN LA ROCHE 2012-10-31 CN disclosed