SCHEMBL28056815

SCHEMBL28056815

O=Cc1cn(CCc2ccccc2)nn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.51
KDM4E B2RXH2 1/20 0.47
KDM6B O15054 1/20 0.47
KDM4A O75164 1/20 0.47
KDM5C P41229 1/20 0.47
KDM4C Q9H3R0 1/20 0.47
KDM2A Q9Y2K7 1/20 0.47
KDM3A Q9Y4C1 1/20 0.47
GBA1 P04062 1/20 0.46
PTGS2 P35354 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4959659 0.83 CYP19A1 (0.56) P2RX7HRH4NPC1RAB9ACYP19A1
SCHEMBL28660008 0.76 HDAC2 (0.48) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL28621784 0.76 HDAC2 (0.48) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL28060209 0.75 HDAC1 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8621793 0.75 GBA1 (0.49) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL16906517 0.75 MAOB (0.51) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL16401668 0.75 GBA1 (0.52) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL17336926 0.74 KDM4E (0.60) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL24569915 0.74 P2RX7 (0.42) P2RX7GBA1
SCHEMBL4964421 0.74 HSP90AB1 (0.52) P2RX7KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096211-B Preparation method of polysubstituted triazole derivative 华侨大学 2021-11-23 CN disclosed
CN-109096211-A A kind of preparation method of polysubstituted triazole derivatives 华侨大学 2018-12-28 CN disclosed
CN-105439966-A Compounds, and preparation method and application thereof UNIV HUAZHONG 2016-03-30 CN disclosed