SCHEMBL8621793

SCHEMBL8621793

Sc1cn(CCc2ccccc2)nn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.49
MAOB P27338 1/20 0.48
MAOA P21397 1/20 0.47
KDM4E B2RXH2 1/20 0.47
KDM6B O15054 1/20 0.47
KDM4A O75164 1/20 0.47
KDM5C P41229 1/20 0.47
KDM4C Q9H3R0 1/20 0.47
KDM2A Q9Y2K7 1/20 0.47
KDM3A Q9Y4C1 1/20 0.47
QPCT Q16769 1/20 0.46
QPCTL Q9NXS2 1/20 0.46
PTGS2 P35354 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521784 0.81 CYP19A1 (0.61) NPC1RAB9AHRH4CYP19A1
SCHEMBL16401668 0.79 GBA1 (0.52) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL16906517 0.79 MAOB (0.51) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL13573675 0.77 PTGS2 (0.70) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL16206231 0.76 GBA1 (0.60) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL27777026 0.76 GBA1 (0.57) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL12853136 0.76 MAOB (0.59) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL28056733 0.75 MAOB (0.48) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL28056815 0.75 P2RX7 (0.51) GBA1MAOBMAOAKDM4EKDM6B
SCHEMBL16903656 0.75 MAOB (0.48) GBA1MAOBMAOAKDM4EKDM6B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842158-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AG (DE) 1998-05-20 EP claimed
WO-1997005119-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1997-02-13 WO claimed
EP-0842158-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AG (DE) 1998-05-20 EP disclosed
EP-0842158-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AG (DE) 1998-05-20 EP disclosed
WO-1997005119-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1997-02-13 WO disclosed
WO-1997005119-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1997-02-13 WO disclosed