SCHEMBL28056881

SCHEMBL28056881

O=C(Cl)c1cccc(I)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
ALOX15 P16050 2/20 0.43
TSHR P16473 1/20 0.42
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
POLB P06746 1/20 0.33
CYP1A2 P05177 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
P2RX7 Q99572 1/20 0.33
PTPRF P10586 1/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5285030 0.84 ALDH1A1 (0.52) ALDH1A1ALOX15TSHRCES2CES1
SCHEMBL2409184 0.83 TSHR (0.63) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL30991215 0.81 TSHR (0.41) ALDH1A1TSHRMEN1KMT2ATDP1
SCHEMBL27867898 0.80 ALDH1A1 (0.35) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL6367716 0.80 ALDH1A1 (0.45) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL29929330 0.79 ALDH1A1 (0.54) ALDH1A1ALOX15MEN1KMT2ATDP1
SCHEMBL502454 0.79 ALDH1A1 (0.54) ALDH1A1ALOX15MEN1KMT2ATDP1
SCHEMBL27841955 0.78 ALDH1A1 (0.43) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL4924666 0.78 ALDH1A1 (0.46) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL2658695 0.78 TSHR (0.38) ALDH1A1TSHRMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105518014-B C-aryl glucoside derivative, preparation method and application thereof in medicine 上海研健新药研发有限公司 2018-03-23 CN disclosed
CN-107311992-A C aryl glucosides derivative, its preparation method and its in application pharmaceutically 上海研健新药研发有限公司 2017-11-03 CN disclosed
CN-105518014-A C-aryl glucoside derivative, preparation method and application thereof in medicine JIANGSU HANSOH PHARMACEUTICAL 2016-04-20 CN disclosed