SCHEMBL28057286

SCHEMBL28057286

Cn1nc(C(=O)ON)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.49
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CFTR P13569 1/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31459702 0.85 ALDH1A1 (0.50) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL17940 0.81 PKM (0.49) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL16863576 0.81 GAA (0.52) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL27787731 0.81 PKM (0.51) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL18510 0.80 PKM (0.54) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL16690902 0.80 PKM (0.50) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL24571057 0.78 PKM (0.49) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL31564889 0.77 PKM (0.40) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL18120300 0.75 PKM (0.47) PKMNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL17894247 0.74 ALDH1A1 (0.46) PKMNPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105452241-B Carboxamides derivatives of ((base of pyrimidine 4) epoxide) 1H indoles 1 and application thereof 诺华股份有限公司 2018-01-05 CN disclosed
CN-105452241-A Pyrimidin-4-yl)oxy)-1H-indole-1-carboxamide derivatives and use thereof NOVARTIS AG 2016-03-30 CN disclosed