SCHEMBL28057940

SCHEMBL28057940

N#Cc1ccc(OC=O)c(O)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.39
CXCR2 P25025 4/20 0.38
CXCR1 P25024 2/20 0.38
CA2 P00918 3/20 0.38
CA12 O43570 1/20 0.38
CA3 P07451 1/20 0.38
CA6 P23280 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.37
ALDH1A1 P00352 1/20 0.36
AOX1 Q06278 1/20 0.36
CA1 P00915 2/20 0.35
PTPN11 Q06124 1/20 0.35
MMP3 P08254 1/20 0.34
AR P10275 1/20 0.34
NCEH1 Q6PIU2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28127287 0.86 P4HB (0.39) P4HBCXCR2CXCR1CA2CA12
SCHEMBL20129681 0.79 MRGPRX4 (0.44) CA2PTGDR2ALDH1A1CA1AR
SCHEMBL28120602 0.77 AR (0.54) P4HBALDH1A1AR
SCHEMBL28862653 0.77 AR (0.50) P4HBALDH1A1AR
SCHEMBL388024 0.76 AR (0.51) P4HBCA2ALDH1A1AOX1CA1
SCHEMBL28107055 0.75 AR (0.46) CA2PTGDR2ALDH1A1CA1AR
SCHEMBL16418462 0.75 ALDH1A1 (0.41) CA2CA12CA9CA14ALDH1A1
SCHEMBL28127063 0.75 PTGDR2 (0.38) CA2CA12CA9PTGDR2CA1
Methyl Alcohol SCHEMBL27451617 0.74 AR (0.50) P4HBALDH1A1AOX1AR
SCHEMBL7512633 0.74 CXCR1 (0.40) P4HBCXCR2CXCR1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107383057-B Imidazoles [4,5-e] thiophene [2,3-b] pyridine derivatives and preparation method thereof with the double fluorescent functionals of solid-liquid 中山大学 2019-04-30 CN disclosed
CN-105209449-B Inhibitors of the kynurenine pathway 库拉德夫制药私人有限公司 2019-02-01 CN disclosed
CN-107383057-A Imidazoles [4,5 e] thiophene [2,3 b] pyridine derivatives with the double fluorescent functionals of solid-liquid and preparation method thereof 中山大学 2017-11-24 CN disclosed
CN-105777781-B Thiazole [4,5 e] thiophene [2,3 b] pyridine derivatives with fluorescent functional and preparation method thereof 中山大学 2017-11-10 CN disclosed
CN-105777781-A Thiazole[4,5-e]thiophene[2,3-b]pyridine type derivative with fluorescent function and preparation method thereof 中山大学 2016-07-20 CN disclosed