SCHEMBL28058232

SCHEMBL28058232

O=C(NCc1ccccc1)OBr

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.55
GAA P10253 1/20 0.53
HPGD P15428 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NCEH1 Q6PIU2 1/20 0.53
KMT2A Q03164 3/20 0.52
CYP2C9 P11712 2/20 0.52
MEN1 O00255 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
ALDH1A1 P00352 3/20 0.51
EPHX1 P07099 1/20 0.50
ALOX12 P18054 1/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19716546 0.82 PLAU (0.54) BCHEGAAHPGDNCEH1KMT2A
SCHEMBL1720194 0.82 ALDH1A1 (0.67) BCHEGAAHPGDSMN1; SMN2KMT2A
SCHEMBL8621389 0.82 GAA (0.55) BCHEGAAHPGDSMN1; SMN2KMT2A
SCHEMBL21201600 0.80 GAA (0.53) BCHEGAAHPGDKMT2ACYP2C9
SCHEMBL29244564 0.80 GAA (0.53) BCHEGAAHPGDKMT2ACYP2C9
SCHEMBL1129046 0.80 CYP2D6 (0.56) BCHEGAAHPGDKMT2ACYP2C9
SCHEMBL2095021 0.80 GAA (0.53) BCHEGAAHPGDSMN1; SMN2KMT2A
SCHEMBL25166809 0.79 CYP1A2 (0.53) BCHEGAASMN1; SMN2CYP1A2CYP2D6
SCHEMBL28053180 0.79 MMP13 (0.55) HPGDSMN1; SMN2ALDH1A1LMNA
SCHEMBL17552096 0.78 NPC1 (0.69) GAAHPGDNCEH1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109136974-A One kind (sp containing C2)-N key compound preparation method 中国科学院上海有机化学研究所 2019-01-04 CN disclosed
CN-108135850-A MODULAR COMPOSITIONS FOR SCAVENGING SOLUBLE BIOMOLECULES AND METHODS RELATED THERETO 纳米提克斯有限责任公司 2018-06-08 CN disclosed
CN-105849099-A Polycyclic inhibitors of cyclin-dependent kinase 7 (CDK7) 达纳-法伯癌症研究所股份有限公司 2016-08-10 CN disclosed
CN-105793262-A Bicyclic alkyne derivatives and uses thereof 新加坡科技研究局 2016-07-20 CN disclosed