SCHEMBL28058540

SCHEMBL28058540

c1cncc(-c2cn[nH]n2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 8/20 1.00
SIRT3 Q9NTG7 1/20 1.00
IDO1 P14902 7/20 0.64
KEAP1 Q14145 1/20 0.64
CYP2A6 P11509 4/20 0.55
ALDH1A1 P00352 3/20 0.55
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
TP53 P04637 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HSD17B10 Q99714 1/20 0.52
ALK Q9UM73 1/20 0.51
METAP1 P53582 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29539786 1.00 METAP2 (1.00) METAP2SIRT3IDO1KEAP1CYP2A6
Ethoxycarbonyl Group SCHEMBL28058501 0.82 METAP2 (0.68) METAP2SIRT3IDO1KEAP1CYP2A6
SCHEMBL8221447 0.79 METAP2 (1.00) METAP2SIRT3IDO1KEAP1METAP1
SCHEMBL5025520 0.77 IDO1 (1.00) METAP2SIRT3IDO1KEAP1METAP1
SCHEMBL8664138 0.77 METAP2 (0.95) METAP2SIRT3IDO1KEAP1METAP1
SCHEMBL29419014 0.72 CYP2A6 (1.00) CYP2A6ALDH1A1CYP1A2CYP3A4KDM4E
SCHEMBL30473120 0.72 CYP2A6 (1.00) CYP2A6ALDH1A1CYP1A2CYP3A4KDM4E
SCHEMBL120088 0.72 CYP2A6 (1.00) CYP2A6ALDH1A1CYP1A2CYP3A4KDM4E
SCHEMBL446537 0.72 METAP2 (0.56) METAP2SIRT3CYP2A6ALDH1A1CYP1A2
SCHEMBL29960290 0.72 METAP2 (0.56) METAP2SIRT3CYP2A6ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105541796-A Synthetic method of NH-1,2,3-triazole bipyridine compounds WUHAN INST TECHNOLOGY 2016-05-04 CN disclosed