SCHEMBL28058828

SCHEMBL28058828

CC(C)(C)C(=O)ON1CCN(CC(F)(F)F)CC1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27600871 0.79 BACE1 (0.34) OPRM1OPRD1OPRK1
SCHEMBL27601011 0.77
SCHEMBL27998224 0.77 ALDH1A1 (0.37)
SCHEMBL27997972 0.77 PAOX (0.40)
SCHEMBL28278579 0.76 KDM4E (0.43)
SCHEMBL28313687 0.76 PRKCQ (0.33)
SCHEMBL27721167 0.76 ALOX15 (0.45)
SCHEMBL28025114 0.76 BACE1 (0.32)
SCHEMBL28869566 0.75 PLA2G10 (0.35)
SCHEMBL28757473 0.75 USP2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-A Quinazolinones PARP-1 inhibitor and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2019-08-02 CN disclosed
CN-106232584-B As 6 inhibitor of histone deacetylase new compound and include its pharmaceutical composition 株式会社钟根堂 2019-06-28 CN disclosed
CN-106232584-A As the new compound of histone deacetylase 6 inhibitor and the pharmaceutical composition comprising it 株式会社钟根堂 2016-12-14 CN disclosed
CN-106187838-A Arylalkyne hydrocarbon compound and its production and use 广东东阳光药业有限公司 2016-12-07 CN disclosed
CN-105461697-A Quinazolinone PARP-1 inhibitors, medicinal composition containing inhibitors, and antitumor use of inhibitors INST MATERIA MEDICA CAMS 2016-04-06 CN disclosed