SCHEMBL28059586

SCHEMBL28059586

NC(C#CC1CCCCC1)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.41
SLC6A2 P23975 2/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAOA P21397 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CYP2A6 P11509 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
FFAR1 O14842 2/20 0.38
FFAR4 Q5NUL3 2/20 0.38
CYP1A2 P05177 1/20 0.37
GRM5 P41594 1/20 0.37
ANPEP P15144 3/20 0.37
CYP2D6 P10635 1/20 0.37
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5966181 0.70 CYP1A2 (0.46) EPHX1TAAR1FFAR1FFAR4CYP1A2
SCHEMBL10716724 0.70 DPP4 (0.49) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL3289204 0.70 DPP4 (0.49) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL131351 0.70 SLC6A2 (0.54) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL3285405 0.68 EPHX1 (0.50) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL27837801 0.68 EPHX1 (0.50) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL3393241 0.68 EPHX1 (0.50) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL10890023 0.68 EPHX1 (0.45) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL28853816 0.68 EPHX1 (0.45) EPHX1SLC6A2TAAR1MAOASLC6A4
SCHEMBL2800708 0.68 ALDH1A1 (0.47) EPHX1CYP1A2GRM5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105481699-B A kind of method for synthesizing the propargylamine derivative for containing different substituents at alkynes end 复旦大学 2017-12-01 CN disclosed
CN-105481699-A Method for synthesizing propargylamine derivative with different substituent groups at alkyne terminal UNIV FUDAN 2016-04-13 CN disclosed