SCHEMBL752316

SCHEMBL752316

O=C(O)N1CC2(CC2)CC1c1ncc(-c2ccc(Br)cc2)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
PRCP P42785 8/20 0.40
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
PDF Q9HBH1 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2707653 0.84 HPGDS (0.42) MAPK13MAPK12MAPK11MAPK14PRCP
SCHEMBL203907 0.84 HPGDS (0.42) MAPK13MAPK12MAPK11MAPK14PRCP
SCHEMBL206727 0.83 ADAM10 (0.42) MAPK13MAPK12MAPK11MAPK14PRCP
SCHEMBL2707006 0.83 ADAM10 (0.42) MAPK13MAPK12MAPK11MAPK14PRCP
SCHEMBL3477648 0.83 CYP3A4 (0.52) PRCPNR1I2ABCB11CYP3A4CYP2C9
SCHEMBL204930 0.82 CYP3A4 (0.40) PRCPNR1I2ABCB11CYP3A4CYP2C9
SCHEMBL19339456 0.81 CYP3A4 (0.43) MAPK13MAPK12MAPK11MAPK14PRCP
SCHEMBL15586557 0.79 CYP3A4 (0.64) PRCPNR1I2ABCB11CYP3A4CYP2C9
SCHEMBL204761 0.79 CYP3A4 (0.64) PRCPNR1I2ABCB11CYP3A4CYP2C9
SCHEMBL2707003 0.79 CYP3A4 (0.64) PRCPNR1I2ABCB11CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed