SCHEMBL28060132

SCHEMBL28060132

O=Cc1ccn(CCc2cccc(OC(F)(F)F)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.50
CHRM1 P11229 1/20 0.50
CHRM3 P20309 1/20 0.50
DAO P14920 1/20 0.44
CNR1 P21554 1/20 0.39
SCD O00767 1/20 0.39
GRM2 Q14416 1/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CETP P11597 1/20 0.38
CARM1 Q86X55 3/20 0.37
PRMT6 Q96LA8 3/20 0.37
MAPK14 Q16539 1/20 0.37
CHRM5 P08912 1/20 0.36
GLS O94925 1/20 0.36
SCN9A Q15858 1/20 0.36
PTGER4 P35408 1/20 0.36
PTGER2 P43116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16347292 0.88 CHRM2 (0.46) CHRM2CHRM1CHRM3DAOSCD
SCHEMBL28060157 0.78 CHRM2 (0.45) CHRM2CHRM1CHRM3DAOCNR1
SCHEMBL5537502 0.73 CHRM2 (0.62) CHRM2CHRM1CHRM3DAOCNR1
SCHEMBL1035570 0.71 CHRM2 (0.58) CHRM2CHRM1CHRM3DAOCNR1
SCHEMBL1047406 0.71 CHRM2 (0.58) CHRM2CHRM1CHRM3DAOCNR1
SCHEMBL2090446 0.71 CHRM2 (0.59) CHRM2CHRM1CHRM3DAOCNR1
SCHEMBL29394922 0.70 PIM1 (0.52) CHRM2CHRM1CHRM3
SCHEMBL68710 0.70 PIM1 (0.52) CHRM2CHRM1CHRM3
SCHEMBL31395106 0.70 MRGPRX4 (0.56) CHRM2CHRM1CHRM3CYP19A1CYP11B1
SCHEMBL5543404 0.70 CHRM2 (0.58) CHRM2CHRM1CHRM3DAOCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492429-A Heteroaryl inhibitors of SUMO activating enzyme MILLENNIUM PHARM INC 2016-04-13 CN disclosed