SCHEMBL28060157

SCHEMBL28060157

CC(=O)Oc1ccn(CCc2cccc(OC(F)(F)F)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
GLS O94925 2/20 0.44
SCD O00767 1/20 0.43
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
CNR1 P21554 1/20 0.42
DAO P14920 1/20 0.41
FLT1 P17948 1/20 0.40
KDR P35968 1/20 0.40
MAPK14 Q16539 1/20 0.39
AMPD2 Q01433 1/20 0.39
GRM2 Q14416 1/20 0.39
SLC6A9 P48067 1/20 0.38
KCNH2 Q12809 1/20 0.38
CETP P11597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28060132 0.78 CHRM2 (0.50) CHRM2CHRM1CHRM3GLSSCD
SCHEMBL1714299 0.74 CYP3A4 (0.58) GLS
SCHEMBL27643005 0.74 CHRM2 (0.53) CHRM2CHRM1CHRM3GLSCNR1
SCHEMBL5181367 0.73 CHRM2 (0.56) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL29103739 0.71 ALDH1A1 (0.53) CHRM2CHRM1CHRM3CYP19A1CYP11B1
SCHEMBL27997591 0.70 CHRM2 (0.55) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL11546048 0.70 CHRM2 (0.51) CHRM2CHRM1CHRM3GLSCNR1
SCHEMBL16347284 0.70 SCD (0.52) CHRM3GLSSCDCYP19A1CYP11B1
SCHEMBL1271844 0.69 FFAR1 (0.67) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL6205346 0.69 CHRM2 (0.53) CHRM2CHRM1CHRM3CNR1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492429-A Heteroaryl inhibitors of SUMO activating enzyme MILLENNIUM PHARM INC 2016-04-13 CN disclosed