SCHEMBL28060180

SCHEMBL28060180

CC(OC=O)c1nnc(CNC(=O)OC(C)(C)C)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
GLS O94925 5/20 0.37
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
CA12 O43570 2/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
PDPK1 O15530 1/20 0.35
GFER P55789 2/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CTSK P43235 3/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25063332 0.76 GAA (0.44) KDM4ELMNAGLSCA1CA2
SCHEMBL28813639 0.75 GLS (0.43) KDM4ELMNAGLSCA1CA2
SCHEMBL10042081 0.74 GLS (0.43) KDM4ELMNAGLSCA1CA2
SCHEMBL15248092 0.74 GLS (0.43) KDM4ELMNAGLSCA1CA2
SCHEMBL15945413 0.73 GLS (0.42) KDM4ELMNAGLSCA1CA2
SCHEMBL11455539 0.73 GLS (0.42) KDM4ELMNAGLSCA1CA2
SCHEMBL8056438 0.73 GLS (0.42) KDM4ELMNAGLSCA1CA2
SCHEMBL18633046 0.72 GLS (0.44) KDM4ELMNAGLSCA1CA2
SCHEMBL18605522 0.71 SMN1; SMN2 (0.50) GLSMEN1GAAKMT2APOLB
SCHEMBL15939915 0.68 GLS (0.39) KDM4ELMNAGLSCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103917528-B PYRIMIDINE PDE10 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-04-20 CN disclosed
CN-103917528-A Pyrimidine PDE10 inhibitors MERCK SHARP & DOHME 2014-07-09 CN disclosed