SCHEMBL28813639

SCHEMBL28813639

CC(C)(C)OC(=O)NCc1nnc(CCOC=O)s1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GLS O94925 14/20 0.43
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
KDM4A O75164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25063332 0.81 GAA (0.44) GLSKDM4ELMNAHTTKDM4A
SCHEMBL11455539 0.78 GLS (0.42) GLSKDM4ELMNAHTTKDM4A
SCHEMBL18633046 0.77 GLS (0.44) GLSKDM4ELMNAHTTKDM4A
SCHEMBL15248092 0.76 GLS (0.43) GLSKDM4ELMNAHTTKDM4A
SCHEMBL10042081 0.76 GLS (0.43) GLSKDM4ELMNAHTTKDM4A
SCHEMBL8056438 0.75 GLS (0.42) GLSKDM4ELMNAHTTKDM4A
SCHEMBL15945413 0.75 GLS (0.42) GLSKDM4ELMNAHTTKDM4A
SCHEMBL28060180 0.75 KDM4E (0.38) GLSKDM4ELMNAL3MBTL1CA12
SCHEMBL18605522 0.73 SMN1; SMN2 (0.50) GLSHTT
SCHEMBL27903373 0.72 KDM4E (0.42) KDM4ELMNAHTTKDM4AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103917528-A Pyrimidine PDE10 inhibitors MERCK SHARP & DOHME 2014-07-09 CN disclosed