SCHEMBL28060593

SCHEMBL28060593

CC(C)Oc1c(C=O)ccc(-c2ccc(F)cc2)c1F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.35
ALDH1A3 P47895 1/20 0.34
ALDH1A1 P00352 3/20 0.34
DRD1 P21728 1/20 0.34
PTGS1 P23219 1/20 0.34
MAPT P10636 1/20 0.34
PTGS2 P35354 2/20 0.33
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KDM4E B2RXH2 2/20 0.32
FFAR4 Q5NUL3 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16056008 0.83 ERN1 (0.43) ERN1ALDH1A1PTGS1MAPTSLC6A4
SCHEMBL505506 0.78 PTGS1 (0.42) ERN1ALDH1A1PTGS1MAPTPTGS2
SCHEMBL16669880 0.77 ALDH1A1 (0.40) ERN1ALDH1A1DRD1PTGS1MAPT
SCHEMBL16616213 0.76 ERN1 (0.34) ERN1ALDH1A3ALDH1A1MAPTPTGS2
SCHEMBL25319381 0.74 MAPT (0.36) ERN1ALDH1A1DRD1PTGS1MAPT
SCHEMBL30482786 0.74 MAPT (0.36) ERN1ALDH1A1DRD1PTGS1MAPT
SCHEMBL21413070 0.74 ALDH1A3 (0.38) ERN1ALDH1A3ALDH1A1MAPTCYP1A2
SCHEMBL18003978 0.74 ERN1 (0.47) ERN1ALDH1A3ALDH1A1MAPTCYP1A2
SCHEMBL38651684 0.73 ALDH1A3 (0.37) ERN1ALDH1A3MAPTLMNACYP1A2
SCHEMBL18489256 0.73 ALDH1A3 (0.37) ERN1ALDH1A3MAPTCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612158-A Antagonists of somatostatin receptor subtype 5 (sstr5) TAKEDA PHARMACEUTICALS CO 2016-05-25 CN disclosed