SCHEMBL28060895

SCHEMBL28060895

O=C(Cl)/C=C/c1ccncn1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.42
JUN P05412 1/20 0.38
NFKB1 P19838 1/20 0.38
PADI4 Q9UM07 1/20 0.37
GRM4 Q14833 1/20 0.35
EPHX2 P34913 1/20 0.35
HSP90AA1 P07900 2/20 0.34
PFKFB3 Q16875 3/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDR P35968 1/20 0.33
TEK Q02763 1/20 0.33
CYP19A1 P11511 1/20 0.32
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
FAAH O00519 1/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25249689 0.82 KDM4E (0.43) P2RX7JUNNFKB1PADI4HDAC6
SCHEMBL6974319 0.82 KDM4E (0.43) P2RX7JUNNFKB1PADI4HDAC6
SCHEMBL8523153 0.81 CCNC (0.49) P2RX7JUNNFKB1PADI4HSP90AA1
SCHEMBL21055912 0.81 CCNC (0.49) P2RX7JUNNFKB1PADI4HSP90AA1
SCHEMBL24150077 0.77 CCNC (0.42) P2RX7JUNNFKB1PADI4PFKFB3
SCHEMBL16264150 0.75 JUN (0.46) P2RX7JUNNFKB1PADI4HSP90AA1
SCHEMBL15171261 0.74 NPC1 (0.58) PADI4HSP90AA1MAPTKDM4EMEN1
SCHEMBL3349779 0.74 NPC1 (0.58) PADI4HSP90AA1MAPTKDM4EMEN1
SCHEMBL24149768 0.74 APP (0.38) P2RX7JUNNFKB1PADI4EPHX2
SCHEMBL1136418 0.74 JUN (0.69) JUNNFKB1PFKFB3HDAC6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105585544-A Trans-substituted alkene derivative, medicine composition containing same and medical application of trans-substituted alkene derivative XIXI HOSPITAL OF HANGZHOU 2016-05-18 CN disclosed