SCHEMBL21055912

SCHEMBL21055912

NC(=O)/C=C/c1ccncn1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNC P24863 2/20 0.49
CDK8 P49336 2/20 0.49
P2RX7 Q99572 1/20 0.42
HSP90AA1 P07900 2/20 0.39
JUN P05412 1/20 0.38
NFKB1 P19838 1/20 0.38
PADI4 Q9UM07 1/20 0.37
MKNK1 Q9BUB5 1/20 0.34
MAP3K7 O43318 4/20 0.33
TAB1 Q15750 4/20 0.33
PFKFB3 Q16875 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDR P35968 1/20 0.33
TEK Q02763 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523153 1.00 CCNC (0.49) CCNCCDK8P2RX7HSP90AA1JUN
SCHEMBL25249689 0.82 KDM4E (0.43) CCNCCDK8P2RX7JUNNFKB1
SCHEMBL6974319 0.82 KDM4E (0.43) CCNCCDK8P2RX7JUNNFKB1
SCHEMBL28060895 0.81 P2RX7 (0.42) P2RX7HSP90AA1JUNNFKB1PADI4
Acrylamide SCHEMBL27993614 0.78 P2RX7 (0.40) CCNCCDK8P2RX7HSP90AA1MKNK1
SCHEMBL24150077 0.77 CCNC (0.42) CCNCCDK8P2RX7JUNNFKB1
SCHEMBL16264150 0.75 JUN (0.46) P2RX7HSP90AA1JUNNFKB1PADI4
SCHEMBL3733195 0.74 NPC1 (0.58) HSP90AA1PADI4NPC1RAB9A
SCHEMBL1382336 0.74 NPC1 (0.58) HSP90AA1PADI4NPC1RAB9A
SCHEMBL24149768 0.74 APP (0.38) CCNCCDK8P2RX7JUNNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050880-B1 QUINAZOLINE DERIVATIVES FOR THE TREATMENT OF CANCER CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2019-06-19 EP disclosed