SCHEMBL28061559

SCHEMBL28061559

Clc1ccc(Oc2c[c]ccc2CCn2cccn2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.35
SLC6A4 P31645 5/20 0.35
KCNH2 Q12809 3/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MAPT P10636 2/20 0.32
NOTUM Q6P988 1/20 0.32
LMNA P02545 2/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32
THRB P10828 2/20 0.32
PTGS1 P23219 2/20 0.31
PTGS2 P35354 2/20 0.31
SCN9A Q15858 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061549 0.77 DRD2 (0.32) SLC6A2SLC6A3LMNATHRBKMT2A
SCHEMBL13739677 0.73 CA12 (0.42) KCNH2MAPTNOTUMPTGS2GAA
SCHEMBL27483390 0.70 TLR8 (0.36) LMNATHRB
SCHEMBL28531127 0.69 CYP19A1 (0.42) SLC6A4SLC6A2MAPTFNTAFNTB
SCHEMBL7023638 0.67 KMT2A (0.46) MAPTLMNAPSEN1PSEN2APH1B
SCHEMBL9560871 0.63 HTR2A (0.41) HTR2ASLC6A4KCNH2SLC6A2SLC6A3
SCHEMBL1355763 0.63 IDO1 (0.44) MAPTLMNATHRBKDM4EALDH1A1
SCHEMBL1375267 0.63 MAPT (0.42) HTR2ASLC6A4KCNH2SLC6A2SLC6A3
SCHEMBL4901152 0.63 IDO1 (0.44) MAPTLMNATHRBKDM4EALDH1A1
SCHEMBL11653814 0.62 L3MBTL1 (0.46) HTR2ASLC6A4KCNH2SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693645-A FUSED HETEROCYCLIC COMPOUNDS AS SODIUM CHANNEL MODULATORS 吉利德科学公司 2016-06-22 CN disclosed
CN-103649056-B Fused heterocyclic compounds as modulators of ion channels GILEAD SCIENCES, INC. (US) 2016-04-27 CN disclosed