SCHEMBL28062880

SCHEMBL28062880

Cn1cc(C=O)c(F)cc1=O

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.46
IMPDH2 P12268 1/20 0.39
ERN1 O75460 2/20 0.36
CREBBP Q92793 1/20 0.34
MAP2K2 P36507 8/20 0.33
MAP2K1 Q02750 8/20 0.33
ATAD2 Q6PL18 1/20 0.33
ATM Q13315 1/20 0.33
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21475934 0.72 MAP2K2 (0.39) CREBBPMAP2K2MAP2K1ATAD2
SCHEMBL18113362 0.72 PRKDC (0.41) ALDH1A1KDM4EIMPDH2ERN1ATAD2
SCHEMBL20157938 0.71 CREBBP (0.35) CREBBPMAP2K2MAP2K1ATAD2
SCHEMBL20157933 0.71 MAP2K1 (0.39) CREBBPMAP2K2MAP2K1ATAD2
SCHEMBL248719 0.69 ERN1 (0.50) ALDH1A1KDM4EERN1
SCHEMBL12172358 0.68 MAP2K2 (0.39) KDM4ECREBBPMAP2K2MAP2K1ATAD2
SCHEMBL1885143 0.68 ALDH1A1 (0.46) ALDH1A1KDM4EIMPDH2ERN1ATM
SCHEMBL2537941 0.67 ALDH1A1 (0.53) ALDH1A1KDM4EIMPDH2ERN1ATM
SCHEMBL18014683 0.67 ALDH1A1 (0.49) ALDH1A1KDM4EIMPDH2ERN1HTR1D
SCHEMBL24196406 0.67 BRD4 (0.42) CREBBPMAP2K2MAP2K1ATAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105622612-A Aminotetrahydropyran derivative used as dipeptidyl peptidase-IV inhibitor CHENGDU BESS CARREY BIOTECHNOLOGY CO LTD 2016-06-01 CN disclosed