SCHEMBL28064501

SCHEMBL28064501

Cc1c(C(N)=O)n(C)c2c(Cl)cccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.41
MCL1 Q07820 3/20 0.40
KDM4E B2RXH2 2/20 0.38
TSHR P16473 2/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PKM P14618 1/20 0.35
PSMB8 P28062 1/20 0.35
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
MAP2 P11137 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
GAA P10253 1/20 0.35
CD38 P28907 2/20 0.34
AKR1B1 P15121 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064659 0.86 MCL1 (0.50) PRMT5MCL1KDM4ETSHRKMT2A
SCHEMBL28064624 0.81 BTK (0.42) MCL1KDM4ETSHRL3MBTL1EGFR
SCHEMBL6595214 0.73 TSHR (0.64) KDM4ETSHRKMT2AL3MBTL1PKM
SCHEMBL35212204 0.73 TSHR (0.64) KDM4ETSHRKMT2AL3MBTL1PKM
SCHEMBL28828000 0.73 KDM4E (0.37) KDM4ETSHRKMT2APOLBSMN1; SMN2
Hydrochloric Acid SCHEMBL28262758 0.72 TSHR (0.62) KDM4ETSHRKMT2AL3MBTL1PKM
SCHEMBL28208613 0.70 TSHR (0.51) KDM4ETSHRKMT2APOLBSMN1; SMN2
SCHEMBL16381206 0.70 FEN1 (0.49) KDM4ETSHRL3MBTL1EGFRSRC
SCHEMBL16571398 0.70 GPR35 (0.36) MCL1KMT2AL3MBTL1MAP2ALDH1A1
SCHEMBL16571676 0.69 GRM2 (0.41) L3MBTL1MAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555763-A Indole-carboxamide derivatives HOFFMANN LA ROCHE 2016-05-04 CN disclosed