SCHEMBL28064659

SCHEMBL28064659

Cc1c(C(=O)O)n(C)c2c(Cl)cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.50
GPR35 Q9HC97 1/20 0.42
FABP4 P15090 1/20 0.40
RORC P51449 3/20 0.40
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DHODH Q02127 1/20 0.39
KMT2A Q03164 3/20 0.38
PRMT5 O14744 1/20 0.38
TSHR P16473 2/20 0.38
NOTUM Q6P988 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
MT-CO2 P00403 1/20 0.38
LMNA P02545 1/20 0.38
TTR P02766 1/20 0.38
PLA2G1B P04054 1/20 0.38
CYP1A2 P05177 1/20 0.38
PGR P06401 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064501 0.86 PRMT5 (0.41) MCL1KDM4EL3MBTL1KMT2APRMT5
SCHEMBL28064638 0.81 MCL1 (0.47) MCL1GPR35FABP4RORCKDM4E
SCHEMBL23809174 0.78 MCL1 (0.45) MCL1GPR35FABP4KDM4EL3MBTL1
SCHEMBL8692545 0.77 GPR35 (0.42) MCL1GPR35TSHRNOTUMUSP2
SCHEMBL24896372 0.75 GPR35 (0.40) MCL1GPR35FABP4KDM4EL3MBTL1
SCHEMBL19331295 0.74 EGFR (0.45) MCL1RORCKDM4EL3MBTL1DHODH
SCHEMBL28828000 0.74 KDM4E (0.37) KDM4EKMT2ATSHRNOTUMLMNA
SCHEMBL1092586 0.73 KDM4E (0.67) MCL1KDM4EL3MBTL1KMT2ATSHR
SCHEMBL30639179 0.73 KDM4E (0.67) MCL1KDM4EL3MBTL1KMT2ATSHR
SCHEMBL28792536 0.71 HTR2C (0.47) MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555763-A Indole-carboxamide derivatives HOFFMANN LA ROCHE 2016-05-04 CN disclosed