SCHEMBL2806543

SCHEMBL2806543

Cc1cc(C(C)(C)c2ccc(C(=O)O)c(C)c2)ccc1C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 3/20 0.59
RXRA P19793 3/20 0.53
NR1H4 Q96RI1 5/20 0.53
ESR1 P03372 1/20 0.52
TDP1 Q9NUW8 1/20 0.50
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
SRD5A2 P31213 1/20 0.42
USP2 O75604 1/20 0.41
CYP2C19 P33261 1/20 0.41
EPHX2 P34913 1/20 0.41
CYP1A2 P05177 1/20 0.41
MYC P01106 1/20 0.41
RARB P10826 1/20 0.41
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30295343 1.00 RXRB (0.59) RXRBRXRANR1H4ESR1TDP1
SCHEMBL162565 0.88 RXRB (0.69) RXRBRXRANR1H4TDP1SRD5A2
SCHEMBL17908058 0.86 RXRB (0.57) RXRBRXRANR1H4TDP1ALDH1A1
SCHEMBL105948 0.85 TDP1 (0.56) RXRBRXRANR1H4ESR1TDP1
SCHEMBL29441322 0.85 TDP1 (0.56) RXRBRXRANR1H4ESR1TDP1
SCHEMBL29361914 0.85 TDP1 (0.56) RXRBRXRANR1H4ESR1TDP1
SCHEMBL7052040 0.84 CDC25A (0.57) RXRBRXRANR1H4ESR1TDP1
SCHEMBL28191970 0.84 RXRB (0.58) RXRBRXRANR1H4TDP1ALDH1A1
SCHEMBL267196 0.83 TDP1 (0.54) RXRBRXRANR1H4ESR1TDP1
SCHEMBL1098811 0.83 TDP1 (0.54) RXRBRXRANR1H4ESR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B RXRB 1440/4885RXRA 1635/4885NR1H4 3516/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 RXRB 3514/4885RXRA 3275/4885NR1H4 2024/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.