Quinoxaline

Quinoxaline

SCHEMBL28065589

O=S(=O)(O)C(F)(F)F.c1ccc2nccnc2c1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.36
PTPN1 P18031 1/20 0.36
TGFBR1 P36897 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPT P10636 2/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
NPC1 O15118 1/20 0.33
ESR1 P03372 1/20 0.33
TP53 P04637 1/20 0.33
RAB9A P51151 1/20 0.33
PTK2B Q14289 1/20 0.33
TSHR P16473 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL5260404 0.85 ALDH1A1 (0.61) ALDH1A1KDM4EALOX12MAPTSMN1; SMN2
Quinoxaline SCHEMBL4270011 0.84 ALDH1A1 (0.44) ALDH1A1KDM4EL3MBTL1ALOX12MAPT
Quinoline SCHEMBL28462226 0.83 ALDH1A1 (0.59) ALDH1A1KDM4EALOX12MAPTSMN1; SMN2
Quinoline SCHEMBL28462227 0.83 ALDH1A1 (0.59) ALDH1A1KDM4EALOX12MAPTSMN1; SMN2
Phenazine SCHEMBL30542151 0.83 MAPT (0.50) ALDH1A1KDM4EPTPN1L3MBTL1MAPT
Quinoxaline SCHEMBL14717879 0.78 ALDH1A1 (0.39) ALDH1A1KDM4EL3MBTL1MAPTSMN1; SMN2
Dipyridyl SCHEMBL15796588 0.78 KDM4E (0.56) ALDH1A1KDM4EL3MBTL1MAPTSMN1; SMN2
Quinoxaline SCHEMBL28035806 0.77 ALDH1A1 (0.45) ALDH1A1TGFBR1L3MBTL1MAPTHDAC1
Trifluoromethanesulfonic Acid SCHEMBL9026926 0.76 KDM4E (0.41) ALDH1A1KDM4EPTPN1L3MBTL1ALOX12
Acridine SCHEMBL3252417 0.76 ALDH1A1 (0.58) ALDH1A1KDM4EPTPN1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683182-A Biaryl acetamide compounds and methods of use thereof 埃姆比特生物科学公司 2016-06-15 CN disclosed