SCHEMBL28065796

SCHEMBL28065796

Clc1cc2ncccc2nc1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.49
NR4A2 P43354 2/20 0.44
HTT P42858 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 6/20 0.43
DOT1L Q8TEK3 2/20 0.41
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
POLB P06746 1/20 0.38
CCR1 P32246 1/20 0.38
CCR8 P51685 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RPS6KA5 O75582 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
S1PR4 O95977 1/20 0.37
CYP3A4 P08684 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CASP1 P29466 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30903381 0.80 CASP6 (0.52) CASP6NR4A2HTTCYP1A2CYP2C19
SCHEMBL6110081 0.80 HTT (0.47) CASP6NR4A2HTTCYP1A2CYP2C19
SCHEMBL24971013 0.80 CASP6 (0.52) CASP6NR4A2HTTCYP1A2CYP2C19
SCHEMBL29987120 0.77 CASP6 (0.58) CASP6NR4A2HTTALDH1A1DOT1L
SCHEMBL28164395 0.74 TDP1 (0.59) CYP1A2ALDH1A1NPC1RAB9APOLB
SCHEMBL28370443 0.73 CASP6 (0.62) CASP6NR4A2HTTCYP1A2CYP2C19
SCHEMBL29812521 0.73 PDGFRB (0.59) CASP6HTTCYP1A2CYP2C19ALDH1A1
SCHEMBL28244742 0.72 KDM4E (0.46) HTTCYP1A2CYP2C19ALDH1A1L3MBTL1
SCHEMBL1750620 0.71 CASP6 (0.71) CASP6NR4A2HTTCYP1A2CYP2C19
SCHEMBL20272948 0.70 ALDH1A1 (0.54) CASP6NR4A2HTTCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102007125-B fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2016-05-25 CN disclosed