SCHEMBL28067942

SCHEMBL28067942

c1ccc(Cc2cccc(C(c3ccccc3)(c3ccccc3)n3ccnc3)c2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 5/20 0.69
CYP11B2 P19099 5/20 0.69
CYP19A1 P11511 6/20 0.52
CYP3A4 P08684 3/20 0.52
NR1I2 O75469 2/20 0.52
ADORA3 P0DMS8 2/20 0.52
TBXA2R P21731 2/20 0.52
CCKBR P32239 2/20 0.52
OPRK1 P41145 2/20 0.52
SLC6A3 Q01959 2/20 0.52
KCNH2 Q12809 2/20 0.52
NR1H4 Q96RI1 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2D6 P10635 2/20 0.52
MAPT P10636 2/20 0.52
TBXAS1 P24557 2/20 0.52
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
SLC22A1 O15245 1/20 0.52
KCNN4 O15554 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL332630 0.83 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL5445913 0.79 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL9720834 0.79 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL8184195 0.79 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL5290299 0.79 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL7159462 0.79 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL28706403 0.79 CYP11B1 (0.67) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL8306981 0.79 CYP11B1 (0.61) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
Hydrochloric Acid SCHEMBL5287102 0.78 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2
SCHEMBL12199510 0.78 CYP11B1 (0.89) CYP11B1CYP11B2CYP19A1CYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108864102-A ERK inhibitor and application method 库拉肿瘤学公司 2018-11-23 CN disclosed
CN-105636586-B ERK inhibitors and methods of use 库拉肿瘤学公司 2018-05-29 CN disclosed
CN-105636586-A ERK inhibitors and methods of use ARAXES PHARMA LLC 2016-06-01 CN disclosed