SCHEMBL28068182

SCHEMBL28068182

O=c1[nH]c2ncc(Br)cc2n1CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.51
ADORA2B P29275 1/20 0.51
GRIN1 Q05586 11/20 0.51
GRIN2B Q13224 11/20 0.51
KMT2A Q03164 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CNOT7 Q9UIV1 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 2/20 0.45
RGS12 O14924 2/20 0.45
USP2 O75604 2/20 0.45
MAPT P10636 2/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
PRKCQ Q04759 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17807874 0.86 GRIN1 (0.52) GRIN1GRIN2B
SCHEMBL15999458 0.77 PDE4A (0.44) GRIN1GRIN2BKMT2AMEN1PRKCQ
SCHEMBL20134012 0.77 GRIN1 (0.58) GRIN1GRIN2B
SCHEMBL31008703 0.77 GRIN1 (0.58) GRIN1GRIN2B
SCHEMBL28829341 0.76 ADORA3 (0.51) ADORA3ADORA2BKMT2AL3MBTL1CNOT7
SCHEMBL22516697 0.76 GRIN1 (0.56) GRIN1GRIN2B
SCHEMBL1564239 0.74 GRIN1 (0.55) GRIN1GRIN2B
SCHEMBL1564343 0.74 GRIN1 (0.55) GRIN1GRIN2B
SCHEMBL1563878 0.74 GRIN1 (0.38) GRIN1GRIN2B
SCHEMBL20874771 0.74 GRIN1 (0.56) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693730-A Heteroaryl compounds, compositions thereof, and their use as protein kinase inhibitors 西格诺药品有限公司 2016-06-22 CN disclosed