SCHEMBL28829341

SCHEMBL28829341

O=c1[nH]c2ncc(Br)nc2n1CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.51
ADORA2B P29275 1/20 0.51
MTOR P42345 2/20 0.48
TSHR P16473 4/20 0.46
LMNA P02545 3/20 0.46
RECQL P46063 1/20 0.46
MDM2 Q00987 1/20 0.46
KMT2A Q03164 4/20 0.45
USP2 O75604 3/20 0.45
MEN1 O00255 3/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPT P10636 3/20 0.45
RGS12 O14924 2/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 4/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL974882 0.86 MTOR (0.62) ADORA3MTORTSHRKMT2AMEN1
SCHEMBL28068276 0.83 MTOR (0.62) ADORA3ADORA2BMTOR
SCHEMBL14874599 0.81 ADORA3 (0.48) ADORA3ADORA2BMTORTSHRLMNA
SCHEMBL28068238 0.79 ADORA3 (0.57) ADORA3ADORA2BTSHRLMNAKMT2A
SCHEMBL28068202 0.78 MTOR (0.51) ADORA3ADORA2BMTORTSHRLMNA
SCHEMBL481737 0.78 MTOR (0.79) MTOR
SCHEMBL30328831 0.77 PDE4A (0.44) ADORA3ADORA2BMTORMAPTADORA2A
SCHEMBL481827 0.77 MTOR (0.43) MTORKDM4EALDH1A1HPGD
SCHEMBL28068182 0.76 ADORA3 (0.51) ADORA3ADORA2BKMT2AUSP2MEN1
SCHEMBL481723 0.75 GRIN1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693730-A Heteroaryl compounds, compositions thereof, and their use as protein kinase inhibitors 西格诺药品有限公司 2016-06-22 CN disclosed