SCHEMBL28068633

SCHEMBL28068633

O=C(CCO)Nc1cccnc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.68
HDAC4 P56524 2/20 0.68
HDAC1 Q13547 2/20 0.68
HDAC7 Q8WUI4 2/20 0.68
HDAC2 Q92769 2/20 0.68
HDAC10 Q969S8 2/20 0.68
HDAC11 Q96DB2 2/20 0.68
HDAC8 Q9BY41 2/20 0.68
HDAC6 Q9UBN7 2/20 0.68
HDAC9 Q9UKV0 2/20 0.68
HDAC5 Q9UQL6 2/20 0.68
POLB P06746 2/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
LMNA P02545 1/20 0.66
EPHX2 P34913 1/20 0.64
PKM P14618 3/20 0.61
NOTUM Q6P988 2/20 0.61
ALDH1A1 P00352 2/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
GAA P10253 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3913781 0.86 HDAC3 (0.68) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL15480449 0.86 HDAC3 (0.88) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3798756 0.86 ALDH1A1 (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5142691 0.85 ALDH1A1 (0.73) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5356584 0.85 SMN1; SMN2 (0.73) HDAC3HDAC4HDAC1HDAC7HDAC2
Iodide SCHEMBL3088158 0.85 HDAC3 (0.66) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8278813 0.85 LMNA (0.78) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28030360 0.83 SMN1; SMN2 (0.67) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL25154931 0.82 HDAC3 (0.71) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1520172 0.82 HDAC3 (0.71) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103687860-B As P2X7Heterocyclic amide derivatives of receptor antagonists 埃科特莱茵药品有限公司 2016-06-08 CN claimed
CN-103687860-B As P2X7Heterocyclic amide derivatives of receptor antagonists 埃科特莱茵药品有限公司 2016-06-08 CN disclosed