SCHEMBL28069299

SCHEMBL28069299

Cc1ccc2c(c1Sc1ccncc1)C(=O)CC(N)=N2

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TYMS P04818 15/20 0.45
DHFR P00374 2/20 0.37
DDAH1 O94760 1/20 0.33
NOS1 P29475 1/20 0.33
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
AURKB Q96GD4 1/20 0.31
INCENP Q9NQS7 1/20 0.31
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30
CDC7 O00311 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27575103 0.70 TYMS (0.40) TYMSDHFRDDAH1NOS1
Hydrochloric Acid SCHEMBL27809309 0.67 TYMS (0.45) TYMSDHFRDDAH1NOS1PDE3B
Nolatrexed SCHEMBL710461 0.62 TYMS (1.00) TYMSDHFR
Nolatrexed SCHEMBL18489 0.62 TYMS (0.66) TYMSDHFR
Nolatrexed SCHEMBL316632 0.62 TYMS (0.97) TYMSDHFR
Nolatrexed SCHEMBL29420099 0.62 TYMS (0.97) TYMSDHFR
SCHEMBL16807869 0.62 TYMS (0.61) TYMSDHFR
Nolatrexed SCHEMBL27935384 0.62 TYMS (0.97) TYMSDHFR
SCHEMBL20434229 0.59 UCHL1 (0.39) TYMS
Hydrochloric Acid SCHEMBL4539745 0.59 TYMS (0.52) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646445-A 2-amino quinazolinone compound synthesis process 吕艳 2016-06-08 CN disclosed