SCHEMBL2806930

SCHEMBL2806930

COCCOc1cc(C=NO)nc2c1ccc1cccnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
ALDH1A1 P00352 3/20 0.40
HSP90AA1 P07900 2/20 0.39
LMNA P02545 7/20 0.39
MAPT P10636 7/20 0.39
KDM4E B2RXH2 5/20 0.38
SMN1; SMN2 Q16637 5/20 0.38
GAA P10253 3/20 0.38
MAPK1 P28482 2/20 0.38
POLB P06746 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
CCR1 P32246 2/20 0.36
CCR5 P51681 2/20 0.36
CCR8 P51685 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2806927 1.00 MEN1 (0.40) MEN1KMT2AALDH1A1HSP90AA1LMNA
SCHEMBL2808443 0.88 KDM4E (0.39) MEN1KMT2AALDH1A1HSP90AA1LMNA
SCHEMBL2808446 0.88 KDM4E (0.39) MEN1KMT2AALDH1A1HSP90AA1LMNA
SCHEMBL2808539 0.87 MAPT (0.41) MEN1KMT2AALDH1A1HSP90AA1LMNA
SCHEMBL2808536 0.87 MAPT (0.41) MEN1KMT2AALDH1A1HSP90AA1LMNA
SCHEMBL2808345 0.87 HSP90AA1 (0.45) MEN1KMT2AHSP90AA1LMNAMAPT
SCHEMBL2808343 0.87 HSP90AA1 (0.45) MEN1KMT2AHSP90AA1LMNAMAPT
SCHEMBL2810871 0.85 MAPT (0.35) KMT2AHSP90AA1LMNAMAPTKDM4E
SCHEMBL2810868 0.85 MAPT (0.35) KMT2AHSP90AA1LMNAMAPTKDM4E
SCHEMBL2805108 0.85 RAB9A (0.43) MEN1KMT2AALDH1A1HSP90AA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140011835-A1 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES NOSCIRA, S.A. (ES) 2014-01-09 US claimed
EP-2002863-A1 [1,10]-phenanthroline derivatives for the treatment of neurodegenerative or haematological diseases NOSCIRA, S.A. (ES) 2008-12-17 EP claimed
US-20140011835-A1 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES NOSCIRA, S.A. (ES) 2014-01-09 US disclosed
US-8592446-B2 [1,10]-phenanthroline derivatives for the treatment of neurodegenerative or haematological diseases NOSCIRA, S.A. (ES) 2013-11-26 US disclosed
US-20100240692-A1 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES NOSCIRA, S.A. (ES) 2010-09-23 US disclosed
EP-2170464-A2 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES NOSCIRA, S.A. (ES) 2010-04-07 EP disclosed
WO-2008152068-A2 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES NOSCIRA, S.A. (ES) 2008-12-18 WO disclosed
EP-2002863-A1 [1,10]-phenanthroline derivatives for the treatment of neurodegenerative or haematological diseases NOSCIRA, S.A. (ES) 2008-12-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140011835-A1 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES HTT, PARK7, ATXN10 MEN1 477/4885KMT2A 250/4885ALDH1A1 319/4885
US-20100240692-A1 [1,10]-PHENANTHROLINE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE OR HAEMATOLOGICAL DISEASES HTT, ATXN10, PSEN1 MEN1 560/4885KMT2A 391/4885ALDH1A1 1502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.