SCHEMBL28069310

SCHEMBL28069310

NC(=O)CNc1ccnc2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.63
ADRA1D P25100 2/20 0.63
ADRA1A P35348 2/20 0.63
ADRA1B P35368 2/20 0.63
FERMT2 Q96AC1 1/20 0.60
HDAC6 Q9UBN7 2/20 0.54
PTPN1 P18031 1/20 0.52
PTPN11 Q06124 1/20 0.52
HRH3 Q9Y5N1 3/20 0.48
DNMT1 P26358 2/20 0.48
HDAC3 O15379 1/20 0.48
ACHE P22303 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
DNMT3L Q9UJW3 1/20 0.48
DNMT3A Q9Y6K1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29362282 0.86 HTR1A (0.65) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL1520512 0.86 HTR1A (0.65) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL6984768 0.82 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL1902196 0.80 PTPN1 (0.67) HTR1AADRA1DADRA1AADRA1BFERMT2
Hydrochloric Acid SCHEMBL7369035 0.79 PTPN1 (0.65) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL29162913 0.77 HRH3 (0.57) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL27902526 0.76 CCNC (0.58) HTR1AADRA1DADRA1AADRA1BPLK4
SCHEMBL6698838 0.76 FERMT2 (1.00) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL9591573 0.76 HTR1A (0.80) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL5511988 0.75 MEN1 (0.59) HTR1AADRA1DADRA1AADRA1BHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106156405-A Organic synthetic route design method based on chemical reaction data storehouse 上海网化化工科技有限公司 2016-11-23 CN disclosed
CN-101595217-B Positively charged water-soluble prodrugs of 1H-imidazo [4,5-c ] quinolin-4-amines and related compounds with fast skin penetration rate 于崇曦 2016-06-08 CN disclosed