SCHEMBL28069640

SCHEMBL28069640

CC(C)(C)[Si](Cl)(c1ccccc1)c1ccccc1.CC(C)(C)[Si](Cl)(c1ccccc1)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 1/20 0.34
MAPK1 P28482 1/20 0.33
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
TSHR P16473 3/20 0.32
TAAR1 Q96RJ0 2/20 0.31
ALOX15 P16050 1/20 0.31
SLC6A2 P23975 1/20 0.31
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
LMNA P02545 1/20 0.30
ALOX12 P18054 1/20 0.30
ACHE P22303 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4241 1.00 ESR1 (0.34) ESR1ESR2ALDH1A1CYP3A4MAPK1
SCHEMBL6391397 0.97 ESR1 (0.33) ESR1ESR2ALDH1A1CYP3A4MAPK1
SCHEMBL2492802 0.95 ESR1 (0.32) ESR1ESR2ALDH1A1CYP3A4MAPK1
SCHEMBL9815122 0.93 ESR1 (0.35) ESR1ESR2ALDH1A1CYP3A4MAPK1
SCHEMBL28398399 0.89
SCHEMBL16458730 0.85 MAPT (0.33) ALDH1A1TSHRLMNAALOX12ACHE
SCHEMBL14837511 0.82 TAAR1 (0.34) TAAR1
SCHEMBL12816750 0.81 TP53 (0.39) ALDH1A1MAPK1LMNA
SCHEMBL12815755 0.80 MEN1 (0.30) ALDH1A1
SCHEMBL9812985 0.80 NR1H2 (0.33) NR1H2NR1H3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777864-A Pentacyclic triterpene-peptide conjugate, and preparation method, medicinal composition and use thereof 中国人民解放军军事医学科学院毒物药物研究所 2016-07-20 CN disclosed