SCHEMBL28069840

SCHEMBL28069840

O=C1c2ccccc2C(O)C1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.50
PARP3 Q9Y6F1 1/20 0.44
EDNRB P24530 1/20 0.40
EDNRA P25101 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
HTR2B P41595 1/20 0.39
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
HBB P68871 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
S100A4 P26447 1/20 0.37
POLB P06746 1/20 0.37
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3994733 0.80 CYP2D6 (0.55) CYP2D6PARP3EDNRBEDNRAMAPT
SCHEMBL7952985 0.80 MEN1 (0.41) CYP2D6EDNRBEDNRAMAPTLMNA
SCHEMBL28225291 0.79 EDNRB (0.44) EDNRBEDNRAMAPTLMNACYP1A2
SCHEMBL27818507 0.77 CYP2D6 (0.51) CYP2D6PARP3EDNRBEDNRAMAPT
SCHEMBL29475772 0.76 CYP2D6 (0.51) CYP2D6PARP3EDNRBEDNRAMAPT
SCHEMBL13917747 0.75 CYP2D6 (0.50) CYP2D6PARP3EDNRBEDNRAMAPT
SCHEMBL17262530 0.75 ACHE (0.38) CYP2D6MAPTLMNATP53CYP1A2
SCHEMBL19926520 0.73 MEN1 (0.42) CYP2D6EDNRBEDNRAMAPTLMNA
SCHEMBL15906510 0.73 CYP2D6 (0.47) CYP2D6EDNRBEDNRAMAPTLMNA
SCHEMBL28055493 0.72 EDNRB (0.46) CYP2D6EDNRBEDNRAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110372550-A Aryl ether and application thereof 佩洛通治疗公司 2019-10-25 CN disclosed
CN-105530923-B Aryl ethers and their use 佩洛通治疗公司 2019-07-23 CN disclosed
CN-105530923-A Aryl ethers and their use PELOTON THERAPEUTICS INC 2016-04-27 CN disclosed