SCHEMBL28069901

SCHEMBL28069901

CC(C)(C)OC(=O)NC(CCO)c1cccc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.47
CTSS P25774 3/20 0.47
CTSB P07858 1/20 0.47
AAK1 Q2M2I8 9/20 0.42
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38666123 1.00 CTSK (0.47) CTSKCTSSCTSBAAK1ROCK2
SCHEMBL29423245 1.00 CTSK (0.47) CTSKCTSSCTSBAAK1ROCK2
SCHEMBL16410211 1.00 CTSK (0.47) CTSKCTSSCTSBAAK1ROCK2
SCHEMBL28069976 0.90 CTSK (0.47) CTSKCTSSCTSBAAK1
SCHEMBL16410495 0.90 CTSK (0.47) CTSKCTSSCTSBAAK1
SCHEMBL29676847 0.90 CTSS (0.49) CTSKCTSSCTSBAAK1
SCHEMBL4838536 0.90 CTSS (0.49) CTSKCTSSCTSBAAK1
SCHEMBL4704028 0.90 CTSS (0.49) CTSKCTSSCTSBAAK1
SCHEMBL4838542 0.90 CTSS (0.49) CTSKCTSSCTSBAAK1
SCHEMBL31163370 0.87 CTSS (0.55) CTSKCTSSCTSBAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555766-A Aminomethyl-biaryl derivatives as complement factor D inhibitors and uses thereof NOVARTIS AG 2016-05-04 CN disclosed