SCHEMBL28071019

SCHEMBL28071019

C1CCC(c2noc(N3CCNCC3)n2)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.41
HRH3 Q9Y5N1 2/20 0.41
PDE10A Q9Y233 1/20 0.39
POLB P06746 1/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
USP7 Q93009 1/20 0.38
GPR119 Q8TDV5 2/20 0.38
HRH1 P35367 1/20 0.38
LCAT P04180 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
USP2 O75604 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALOX5AP P20292 1/20 0.36
KCNH2 Q12809 1/20 0.36
PLAT P00750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17115054 0.98 POLB (0.41) HRH4HRH3PDE10APOLBCASP3
SCHEMBL17115090 0.93 PDE10A (0.44) HRH4HRH3PDE10AUSP7GPR119
SCHEMBL12506093 0.82 GPR119 (0.56) POLBCASP3SENP7SENP6GPR119
SCHEMBL12506078 0.81 GPR119 (0.55) POLBCASP3SENP7SENP6GPR119
SCHEMBL19399166 0.80 CHRM3 (0.47) PDE10APOLBCASP3SENP7SENP6
SCHEMBL15312852 0.79 GPR119 (0.56) POLBCASP3SENP7SENP6USP7
SCHEMBL3694402 0.75 GPR119 (0.59) USP7GPR119LCATALOX5AP
SCHEMBL17115089 0.74 HRH4 (0.39) HRH4PDE10AGPR119ALOX5AP
SCHEMBL19454413 0.73 GPR119 (0.46) POLBUSP7GPR119LCATSMN1; SMN2
SCHEMBL1103825 0.73 CHRM3 (0.44) PDE10AUSP7GPR119LCATALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646492-A Five-membered-aromatic-heterocycte-containing substituted xanthine compound and preparation method and use thereof 中国医学科学院药物研究所 2016-06-08 CN disclosed