SCHEMBL15312852

SCHEMBL15312852

OC1CCN(c2nc(C3CCC3)no2)CC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.56
LCAT P04180 1/20 0.42
ALOX5AP P20292 5/20 0.40
CHRM3 P20309 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
POLB P06746 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP7 Q93009 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12506093 0.97 GPR119 (0.56) GPR119LCATALOX5APCHRM3PDE4A
SCHEMBL12506078 0.95 GPR119 (0.55) GPR119LCATALOX5APCHRM3PDE4A
SCHEMBL3694402 0.93 GPR119 (0.59) GPR119LCATALOX5APCHRM3PDE4A
SCHEMBL19399166 0.81 CHRM3 (0.47) GPR119LCATCHRM3PDE4APDE4B
SCHEMBL28071019 0.79 HRH4 (0.41) GPR119LCATALOX5APPOLBCASP3
SCHEMBL19454413 0.78 GPR119 (0.46) GPR119LCATCHRM3PDE4APDE4B
SCHEMBL17115054 0.78 POLB (0.41) GPR119LCATALOX5APPOLBCASP3
SCHEMBL1103825 0.78 CHRM3 (0.44) GPR119LCATALOX5APCHRM3PDE4A
SCHEMBL13404980 0.76 GPR119 (0.64) GPR119ALOX5APCHRM3PDE4APDE4B
SCHEMBL17115090 0.75 PDE10A (0.44) GPR119LCATALOX5APCHRM3PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8853213-B2 Bicyclic compound for modulating G protein-coupled receptors HANMI PHARM. CO., LTD (KR) 2014-10-07 US disclosed
US-20130274268-A1 NEW BICYCLIC COMPOUND FOR MODULATING G PROTEIN-COUPLED RECEPTORS HANMI PHARM. CO., LTD (KR) 2013-10-17 US disclosed
CN-103328482-A New bicyclic compound for modulating G protein-coupled receptors HANMI PHARM IND CO LTD 2013-09-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130274268-A1 NEW BICYCLIC COMPOUND FOR MODULATING G PROTEIN-COUPLED RECEPTORS GPR119, GPR65, GPR3 GPR119 1/4885LCAT 822/4885ALOX5AP 1813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.