SCHEMBL28071862

SCHEMBL28071862

Nc1cc(-c2ccc(C(F)(F)F)cc2)nc(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.59
ADORA1 P30542 2/20 0.59
ADORA3 P0DMS8 1/20 0.52
KIF11 P52732 2/20 0.47
KDM4E B2RXH2 5/20 0.46
DPP4 P27487 1/20 0.46
LTA4H P09960 1/20 0.45
ALDH1A1 P00352 2/20 0.45
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
TOP1 P11387 2/20 0.44
HRH4 Q9H3N8 1/20 0.43
LMNA P02545 1/20 0.43
THRB P10828 1/20 0.43
BACE1 P56817 1/20 0.42
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3898550 0.94 ADORA2A (0.72) ADORA2AADORA1ADORA3KIF11KDM4E
SCHEMBL3898780 0.92 ADORA2A (0.51) ADORA2AADORA1ADORA3KIF11KDM4E
SCHEMBL22234018 0.91 KIF11 (0.52) ADORA2AADORA1ADORA3KIF11DPP4
SCHEMBL3910159 0.86 ADORA2A (0.53) ADORA2AADORA1ADORA3KIF11KDM4E
SCHEMBL2088245 0.84 KIF11 (0.48) ADORA2AADORA3KIF11KDM4ELTA4H
SCHEMBL29894012 0.83 S1PR1 (0.46) ADORA2AADORA1ADORA3KIF11KDM4E
SCHEMBL29893642 0.83 KDM4E (0.46) ADORA2AADORA1ADORA3KIF11KDM4E
SCHEMBL6531140 0.82 ADORA2A (0.54) ADORA2AADORA1ADORA3KDM4EALDH1A1
SCHEMBL1257904 0.81 KIF11 (0.56) ADORA3KIF11KDM4EDPP4LTA4H
SCHEMBL6528840 0.81 S1PR1 (0.54) KDM4EALDH1A1MEN1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683166-A Substituted pyrimidine Bmi-1 inhibitors PTC医疗公司 2016-06-15 CN disclosed