Ergocryptine

Ergocryptine

SCHEMBL28072302

CC(C)CC1C(=O)N2CCCC2C2(O)OC(NC(=O)C3C=C4c5cccc6[nH]cc(c56)CC4N(C)C3)(C(C)C)C(=O)N12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 1.00
MAPT P10636 10/20 1.00
CYP3A4 P08684 9/20 1.00
MEN1 O00255 8/20 1.00
KMT2A Q03164 8/20 1.00
ALDH1A1 P00352 7/20 1.00
CYP2C9 P11712 7/20 1.00
HIF1A Q16665 7/20 1.00
ABCB1 P08183 7/20 1.00
HPGD P15428 5/20 1.00
USP2 O75604 5/20 1.00
LMNA P02545 5/20 1.00
ADRA2A P08913 5/20 1.00
DRD1 P21728 5/20 1.00
DRD3 P35462 5/20 1.00
HSD17B10 Q99714 4/20 1.00
CYP2C19 P33261 4/20 1.00
NPSR1 Q6W5P4 4/20 1.00
DRD2 P14416 4/20 1.00
ADRA2B P18089 4/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ergocryptine SCHEMBL30498875 1.00 KDM4E (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocryptine SCHEMBL29372991 1.00 KDM4E (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocryptine SCHEMBL29376491 1.00 KDM4E (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocryptine SCHEMBL78951 1.00 KDM4E (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocryptine SCHEMBL11034170 1.00 KDM4E (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocryptine SCHEMBL12481541 0.98 KDM4E (0.95) KDM4EMAPTCYP3A4MEN1KMT2A
SCHEMBL30449023 0.94 MAPT (0.88) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocristine SCHEMBL29386896 0.93 MAPT (0.89) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocristine SCHEMBL30957132 0.92 CYP2C9 (1.00) KDM4EMAPTCYP3A4MEN1KMT2A
Ergocristine SCHEMBL14029486 0.92 CYP2C9 (1.00) KDM4EMAPTCYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118209655-A Method for detecting ergot alkaloid in food 安徽省疾病预防控制中心(省健康教育所、省公共卫生研究院) 2024-06-18 CN disclosed
CN-112521407-B Preparation of bromocriptine mesylate 天津康哲医药科技发展有限公司 2022-08-05 CN disclosed
CN-112521407-A Preparation of bromocriptine mesylate 天津康哲医药科技发展有限公司 2021-03-19 CN disclosed
CN-105560244-B A kind of inhibitors of gamma-secretase and its application 上海交通大学 2019-01-11 CN disclosed
CN-105560244-A Gamma-secretase inhibitor and use thereof UNIV SHANGHAI JIAOTONG 2016-05-11 CN disclosed