SCHEMBL28073682

SCHEMBL28073682

O=C(N=[N+]=Nc1ccc(-n2nc(C3CC3)cc2C2CC2)cc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRACR2A Q9BSW2 9/20 0.51
ORAI1 Q96D31 4/20 0.43
KCNJ6 P48051 4/20 0.38
KCNJ3 P48549 4/20 0.38
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KCNJ5 P48544 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28950389 0.86 CRACR2A (0.43) CRACR2AORAI1
SCHEMBL1667966 0.74 CRACR2A (0.81) CRACR2AORAI1KCNJ6KCNJ3
SCHEMBL1671385 0.70 CRACR2A (0.55) CRACR2AORAI1KCNJ6KCNJ3NPC1
SCHEMBL28106553 0.68 CES2 (0.46) NPC1LMNAPKMRAB9ASMN1; SMN2
SCHEMBL1671387 0.67 CRACR2A (1.00) CRACR2AORAI1NPC1RAB9ASMN1; SMN2
SCHEMBL28065979 0.67 CES2 (0.47) NPC1LMNARAB9ASMN1; SMN2
SCHEMBL27563970 0.66 CCNA2 (0.36) NPC1RAB9ASMN1; SMN2
SCHEMBL1879322 0.66 CRACR2A (0.67) CRACR2AORAI1KCNJ6KCNJ3LMNA
SCHEMBL1666818 0.65 CRACR2A (0.58) CRACR2AORAI1LMNAPKM
Hydrochloric Acid SCHEMBL1668379 0.65 CRACR2A (0.75) CRACR2AORAI1NPC1TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102834382-B The pyrazole derivatives of calcium channel modulators is activated as calcium release 理森制药股份公司 2016-08-03 CN claimed
CN-102834382-B The pyrazole derivatives of calcium channel modulators is activated as calcium release 理森制药股份公司 2016-08-03 CN disclosed