SCHEMBL28074404

SCHEMBL28074404

O=C(O)C1CCc2c(c3cc(OCc4ccccc4)ccc3n2Cc2ccc(F)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 4/20 0.50
EGFR P00533 2/20 0.50
IGF1R P08069 2/20 0.50
FLT4 P35916 2/20 0.50
KDR P35968 2/20 0.50
HDAC6 Q9UBN7 3/20 0.48
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 2/20 0.45
AKR1C4 P17516 1/20 0.45
PTGS1 P23219 1/20 0.45
AKR1C1 Q04828 1/20 0.45
EDNRB P24530 2/20 0.45
EDNRA P25101 2/20 0.45
S1PR1 P21453 2/20 0.44
PRKX P51817 1/20 0.44
ACVR1 Q04771 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.44
ENPP2 Q13822 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28074607 0.94 EGFR (0.50) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL28074596 0.92 AKR1C3 (0.54) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL28074399 0.91 HDAC6 (0.49) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL7662475 0.86 EGFR (0.49) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL28074421 0.86 AKR1C3 (0.61) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL28495133 0.85 EDNRB (0.45) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL28503511 0.82 HDAC6 (0.44) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL11836056 0.80 AKR1C3 (0.64) S1PR5EGFRIGF1RFLT4KDR
SCHEMBL9458829 0.79 ALOX5AP (0.59) PTGS1
SCHEMBL28500992 0.79 AKR1C3 (0.74) S1PR5EGFRIGF1RFLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN claimed
CN-105646330-A Heteroaromatic ring derivative and application thereof in drug 贵州医科大学 2016-06-08 CN claimed
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN disclosed
CN-105646330-A Heteroaromatic ring derivative and application thereof in drug 贵州医科大学 2016-06-08 CN disclosed