SCHEMBL28074607

SCHEMBL28074607

O=C(O)C1CCc2c(c3cc(OCc4ccccc4)ccc3n2Cc2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.50
IGF1R P08069 2/20 0.50
FLT4 P35916 2/20 0.50
KDR P35968 2/20 0.50
HDAC6 Q9UBN7 2/20 0.49
AKR1C3 P42330 2/20 0.49
AKR1C2 P52895 2/20 0.49
AKR1C4 P17516 1/20 0.49
PTGS1 P23219 1/20 0.49
AKR1C1 Q04828 1/20 0.49
S1PR5 Q9H228 3/20 0.49
S1PR1 P21453 2/20 0.48
PRKX P51817 1/20 0.48
ACVR1 Q04771 1/20 0.48
PLA2G2A P14555 4/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAPKAPK2 P49137 1/20 0.46
EDNRB P24530 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28074596 0.95 AKR1C3 (0.54) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL28074404 0.94 S1PR5 (0.50) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL28074399 0.94 HDAC6 (0.49) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL7662475 0.91 EGFR (0.49) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL28495133 0.88 EDNRB (0.45) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL11836056 0.85 AKR1C3 (0.64) EGFRIGF1RFLT4KDRAKR1C3
SCHEMBL28503511 0.85 HDAC6 (0.44) EGFRIGF1RFLT4KDRHDAC6
SCHEMBL28500992 0.83 AKR1C3 (0.74) EGFRIGF1RFLT4KDRAKR1C3
SCHEMBL28488499 0.83 AKR1C3 (0.74) EGFRIGF1RFLT4KDRAKR1C3
SCHEMBL28487851 0.83 AKR1C3 (0.74) EGFRIGF1RFLT4KDRAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN claimed
CN-105646330-A Heteroaromatic ring derivative and application thereof in drug 贵州医科大学 2016-06-08 CN claimed
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN disclosed
CN-105646330-A Heteroaromatic ring derivative and application thereof in drug 贵州医科大学 2016-06-08 CN disclosed