SCHEMBL28074771

SCHEMBL28074771

[CH2]Cc1cn(Cc2ccccc2)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.49
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2E1 P05181 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2B6 P20813 1/20 0.48
CYP2C19 P33261 1/20 0.48
CYP19A1 P11511 4/20 0.44
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
KDM4C Q9H3R0 2/20 0.44
KDM5A P29375 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
PHF8 Q9UPP1 1/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
TBXAS1 P24557 1/20 0.44
QPCT Q16769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30741761 0.84 HPGDS (0.50) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL28417084 0.84 HPGDS (0.50) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL8862886 0.83 HTT (0.41) KDM4CKDM5AKDM5BMAPTNPC1
SCHEMBL8794954 0.83 CYP11B1 (0.47) CYP19A1CYP11B1CYP11B2KDM4CKDM5A
SCHEMBL28422539 0.82 HPGDS (0.49) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL28417071 0.82 HPGDS (0.49) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL1187114 0.82 KDM4E (0.50) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL5023714 0.82 HPGDS (0.49) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL9598245 0.82 CYP3A4 (0.51) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6
SCHEMBL6896976 0.79 HPGDS (0.50) HPGDSCYP3A4CYP2D6CYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829317-B Imidazopyrazines ketone derivatives 默克专利股份公司 2019-03-29 CN disclosed
CN-106458988-A Heterocyclyl-butanamide derivatives 默克专利股份公司 2017-02-22 CN disclosed
CN-105829317-A Imidazopyrazinone derivatives 默克专利股份公司 2016-08-03 CN disclosed