SCHEMBL28074783

SCHEMBL28074783

COC(=O)c1ccc2c(c1)NC(=O)C2=Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.58
RAF1 P04049 1/20 0.58
PIM1 P11309 2/20 0.57
PDPK1 O15530 1/20 0.57
RET P07949 3/20 0.54
PLK4 O00444 2/20 0.51
PLK1 P53350 2/20 0.51
PSEN1 P49768 1/20 0.51
PSEN2 P49810 1/20 0.51
APH1B Q8WW43 1/20 0.51
NCSTN Q92542 1/20 0.51
APH1A Q96BI3 1/20 0.51
PSENEN Q9NZ42 1/20 0.51
DHFR P00374 1/20 0.50
JAK3 P52333 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
LRRK2 Q5S007 1/20 0.49
FLT3 P36888 1/20 0.48
PDGFRB P09619 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28655203 0.87 RAF1 (0.59) AURKARAF1PIM1PDPK1PLK4
SCHEMBL14521088 0.85 FLT3 (0.57) AURKARAF1PIM1PDPK1PLK4
SCHEMBL14521057 0.84 PDPK1 (0.54) AURKARAF1PIM1PDPK1PLK4
SCHEMBL14521053 0.83 PDPK1 (0.53) AURKARAF1PIM1PDPK1PLK4
SCHEMBL14521033 0.83 NPC1 (0.60) AURKARAF1PIM1PDPK1RET
SCHEMBL14521087 0.83 PDPK1 (0.55) AURKARAF1PIM1PDPK1PSEN1
SCHEMBL20710199 0.83 PDPK1 (0.49) AURKARAF1PDPK1RETNPC1
SCHEMBL14521098 0.82 NPC1 (0.52) AURKARAF1PIM1PDPK1RET
SCHEMBL14521054 0.82 XDH (0.52) AURKARAF1PIM1PDPK1NPC1
SCHEMBL14521055 0.82 CSNK1D (0.54) AURKARAF1PDPK1RETDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107868087-B Method for preparing pyrroloindole derivatives 浙江大学 2020-03-24 CN disclosed
CN-105837493-A A synthetic method of Nintedanib and an intermediate of Nintedanib 东南大学 2016-08-10 CN disclosed