SCHEMBL28095676

SCHEMBL28095676

COc1ccc(-c2n[nH]c(-c3ccc4c(c3)OCO4)n2)cc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 1/20 0.51
GRK6 P43250 1/20 0.47
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 1/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA1 P30542 1/20 0.44
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28075558 0.86 DCUN1D1 (0.51) DCUN1D1IDO1TDO2NPC1RAB9A
SCHEMBL28095608 0.86 DCUN1D1 (0.51) DCUN1D1IDO1TDO2NPC1RAB9A
SCHEMBL28075557 0.82 GRK6 (0.52) DCUN1D1GRK6NPC1RAB9ASMN1; SMN2
SCHEMBL28096083 0.79 MAPT (0.49) DCUN1D1SMN1; SMN2KDM4EHSD17B10TP53
SCHEMBL17280056 0.79 DCUN1D1 (0.62) DCUN1D1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL28096010 0.78 KDM4E (0.55) GRK6KDM4EHSD17B10POLBTSHR
SCHEMBL18927318 0.76 SMN1; SMN2 (0.56) IDO1TDO2NPC1RAB9ASMN1; SMN2
SCHEMBL28833481 0.74 AMY1A (0.46) GRK6NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL23388700 0.73 DCUN1D1 (0.54) DCUN1D1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL15436211 0.71 KIT (0.58) DCUN1D1IDO1TDO2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed