SCHEMBL28076115

SCHEMBL28076115

NS(=O)(=O)c1cc2cc(-c3cc(Cl)ccc3C[SH](=O)=O)ccc2o1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.45
CA1 P00915 5/20 0.44
CA12 O43570 4/20 0.44
CA9 Q16790 4/20 0.44
CCR2 P41597 2/20 0.36
AKR1B1 P15121 1/20 0.36
NT5E P21589 1/20 0.35
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076116 0.78 CCR2 (0.54) CA2CA1CA12CA9CCR2
SCHEMBL28076323 0.75 CA2 (0.45) CA2CA1CA12CA9CCR2
SCHEMBL28076294 0.75 PTGS1 (0.39)
SCHEMBL28076138 0.68 PTGES2 (0.39) CA2CA1CA12CA9
SCHEMBL28076281 0.66 CCR2 (0.64) CCR2
SCHEMBL28076366 0.65 PTGDR2 (0.41) CA2CA1CA12CA9
SCHEMBL18333467 0.64 CA2 (1.00) CA2CA1CA12CA9
SCHEMBL4483300 0.64 CCR2 (0.54) CA2CA1CA12CA9CCR2
SCHEMBL10506991 0.63 CA2 (0.67) CA2CA1CA12CA9MAOB
SCHEMBL10508948 0.63 CA2 (1.00) CA2CA1CA12CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103380115-B Sulfur derivatives as chemokine receptor modulators 阿勒根公司 2016-08-24 CN claimed
CN-106220618-B Sulfur derivatives as chemokine receptor modulators 阿勒根公司 2019-04-26 CN disclosed
CN-106220618-A SULFUR DERIVATIVES AS CHEMOKINE RECEPTOR MODULATORS 阿勒根公司 2016-12-14 CN disclosed
CN-103380115-B Sulfur derivatives as chemokine receptor modulators 阿勒根公司 2016-08-24 CN disclosed