SCHEMBL28076540

SCHEMBL28076540

Cc1c(-c2ccc(N)nc2)ccnc1Br

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTOR P42345 8/20 0.41
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
PIK3CD O00329 2/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAP4K4 O95819 2/20 0.38
PDE10A Q9Y233 1/20 0.37
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.36
MINK1 Q8N4C8 1/20 0.36
TNIK Q9UKE5 1/20 0.36
TDO2 P48775 2/20 0.36
FEN1 P39748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30522547 0.83 MTOR (0.52) MTORNOS3NOS2PIK3CDMKNK1
SCHEMBL29264261 0.73 LMNA (0.39) KDM4EGAACYP1A2
SCHEMBL14975663 0.73 ALDH1A1 (0.45) KDM4EALDH1A1MAP4K4CYP1A2
SCHEMBL30957760 0.73 LMNA (0.39) KDM4EGAACYP1A2
SCHEMBL16681201 0.72 ABL1 (0.48) MTORNOS3NOS2PIK3CDMKNK1
SCHEMBL30522583 0.71 ALOX5AP (0.47) MTORNOS3NOS2PDE10AFEN1
SCHEMBL15730148 0.69 MKNK1 (0.57) MTORNOS3NOS2PIK3CDMKNK1
SCHEMBL22675252 0.69 CYP3A4 (0.45) NOS3NOS2KDM4EALDH1A1GAA
SCHEMBL3813230 0.69 ABL1 (0.63) NOS3NOS2PIK3CDMKNK1MKNK2
SCHEMBL11072269 0.69 CCNC (0.46) MTORNOS3NOS2PIK3CDMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658646-B Aminoheteroaryl benzamide as kinase inhibitor 诺华股份有限公司 2018-11-27 CN disclosed
CN-105658646-A Aminoheteroaryl benzamides as kinase inhibitors 诺华股份有限公司 2016-06-08 CN disclosed