SCHEMBL28078227

SCHEMBL28078227

Nc1cc[nH]c1-c1ccc(NC(=O)Nc2cc(C(F)(F)F)ccc2F)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CA9 Q16790 1/20 0.60
RIPK1 Q13546 2/20 0.59
FLT3 P36888 6/20 0.58
PDGFRB P09619 4/20 0.58
NTRK1 P04629 3/20 0.58
NTRK2 Q16620 3/20 0.58
RET P07949 2/20 0.58
NTRK3 Q16288 2/20 0.58
AURKB Q96GD4 2/20 0.58
LTK P29376 1/20 0.58
CDK8 P49336 1/20 0.58
MAPK14 Q16539 1/20 0.58
KDR P35968 14/20 0.57
KIT P10721 6/20 0.57
FLT1 P17948 5/20 0.57
CSF1R P07333 4/20 0.57
FLT4 P35916 4/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1924313 0.84 KDR (0.60) CA12CA1CA2CA9RIPK1
SCHEMBL1924576 0.80 CA12 (0.55) CA12CA1CA2CA9RIPK1
SCHEMBL4340395 0.80 CA12 (0.69) CA12CA1CA2CA9RIPK1
Hydrochloric Acid SCHEMBL1924264 0.79 CA12 (0.54) CA12CA1CA2CA9RIPK1
SCHEMBL5241624 0.79 RIPK1 (0.50) RIPK1FLT3PDGFRBNTRK1NTRK2
SCHEMBL21750852 0.78 CA12 (0.70) CA12CA1CA2CA9RIPK1
SCHEMBL4662498 0.78 KDR (0.60) CA12CA1CA2CA9RIPK1
SCHEMBL5264573 0.78 RIPK1 (0.64) CA12CA1CA2CA9RIPK1
SCHEMBL27663136 0.78 CA12 (0.57) CA12CA1CA2CA9RIPK1
SCHEMBL1923687 0.78 CA12 (0.57) CA12CA1CA2CA9RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105732634-A Substituted 4-amino-pyrrolotriazine derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis 拜尔健康护理有限责任公司 2016-07-06 CN disclosed