SCHEMBL28078259

SCHEMBL28078259

Brc1ccc(-c2ccc(-c3ccncn3)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.50
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.44
HDAC4 P56524 1/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPK1 P28482 2/20 0.39
METAP2 P50579 1/20 0.38
MAPK10 P53779 2/20 0.38
MAPK14 Q16539 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
NPC1 O15118 4/20 0.38
NFKB1 P19838 2/20 0.38
NFKB2 Q00653 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566727 0.98 CYP2D6 (0.51) CYP2D6RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL30273511 0.98 CYP2D6 (0.51) CYP2D6RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL9903935 0.87 CYP2D6 (0.60) CYP2D6LMNAHDAC4MAPTMAPK1
SCHEMBL31360692 0.81 NOTUM (0.52) CYP2D6HDAC4MAPTMAPK14MAPK9
SCHEMBL3157652 0.81 NOTUM (0.52) CYP2D6HDAC4MAPTMAPK14MAPK9
SCHEMBL8695286 0.81 CYP2D6 (0.60) CYP2D6RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL8499115 0.80 CYP2D6 (0.53) CYP2D6RAB9ALMNAMAPTMAPK10
SCHEMBL28135256 0.80 MAPK14 (0.40) CYP2D6RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL15651713 0.77 CYP2D6 (0.51) CYP2D6RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL675705 0.77 CYP2D6 (0.51) CYP2D6HDAC4MAPTMAPK1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106397415-A Pyridine-based five-membered-ring substituted compound and application thereof 江苏三月光电科技有限公司 2017-02-15 CN disclosed
CN-105732588-A Organic Compound, Light-Emitting Element, Display Module, Lighting Module, Light-Emitting Device, Display Device, Electronic Device, and Lighting Device 株式会社半导体能源研究所 2016-07-06 CN disclosed